Hart C.J.S., Riches A.G., Tiash S., Clapper E., Ramu S., Zuegg J., Ryan J.H., Skinner-Adams T.S. (2022) Submitted for publication. A subset screen of the Compounds Australia Scaffold Library identifies 7- acylaminodibenzoxazepinones as potent and selective hits for anti-Giardia drug discovery
Riches A.G., Hart C.J.S., Schmit M., Debele E., Tiash S., Clapper E., Skinner-Adams T.S., Ryan J.H., (2022) Submitted for publication. Structural reassignment of a dibenz[b,f][1,4]oxazepin-11(10H)-one with potent antigiardial activity.
Hagan, K.D., Hart C. J. S., McInally, S.G., Dawson, S.C. (2021). In press. Harnessing the power of molecular genetic tools to illuminate Giardia biology and pathogenesis. Current Tropical Medicine Reports.
Riches, A. G., Hart C. J. S., Trenholme, K. R., Skinner-Adams, T. S. (2020). Anti-Giardia Drug Discovery: Current Status and Gut Feelings. Journal of Medicinal Chemistry. DOI: 10.1021/acs.jmedchem.0c00910 Citations: 18
Tiash, S., Saunders, J., Hart, C. J. S., Ryan, J. H., Riches, A. G., Skinner-Adams, T.S. (2020). An image-based Pathogen Box screen identifies new compounds with anti-Giardia activity and highlights the importance of assay choice in phenotypic drug discovery. International Journal for Parasitology: Drugs and Drug Resistance, 12(2020), 60-67. DOI: 10.1016/j.ijpddr.2020.03.002. Citations: 3
Hart, C. J. S., Munro, T., Andrews, K. T., Ryan, J. H., Riches, A. G., & Skinner-Adams, T. S. (2017). A novel in vitro image-based assay identifies new drug leads for giardiasis. International Journal for Parasitology: Drugs and Drug Resistance, 7(1), 83–89. DOI: 10.1016/j.ijpddr.2017.01.005. Citations: 26
Hart, C. Cock, I.E. (2016). An examination of the antimicrobial and anticancer properties of Garcinia cambogia fruit pericarp extracts. BEMS Reports, 2(2), 55–63. DOI: 10.5530/BEMS.2016.2.10. Citations: 21
Hart, C., Ilanko, P., Sirdaarta, J., Rayan, P., McDonnell, P.A., Cock, I.E. (2014). Tasmannia stipitata as a functional food/natural preservative: antimicrobial activity and toxicity. Pharmacognosy communications, 4(4), 33–47. DOI: 10.5530/pc.2014.4.4. Citations: 56